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5

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0395 Pyrantel tartrate

Banminth,酒石酸噻吩嘧啶

Antibiotic; Parasite Microbiology/Virology
Pyrantel tartrate (Banminth) 是一种四氢嘧啶类广谱牲畜驱虫剂,是烟碱乙酰胆碱受体激动剂。它能引起寄生虫的痉挛性肌肉麻痹。它可研究胃肠道线虫感染。
T1259 Pyrantel pamoate

双羟萘酸噻嘧啶,Pyrantel embonate

Others; Antibiotic; Parasite Microbiology/Virology; Others
Pyrantel pamoate (Pyrantel embonate) 是一种四氢嘧啶光谱驱虫剂,是烟碱乙酰胆碱受体激动剂。它可引起寄生虫的痉挛性肌肉麻痹。它可研究胃肠道线虫感染。
T37757 Tyvelose

Tyvelose is an unusual 3,6-dideoxyhexose terminal sugar and the immunodominant component of glycoprotein antigens in the parasitic helminth T. spiralis, which is responsible for trichinosis in humans. It is produced in high amounts by the infective larva and is immunodominant during the muscle stage of infection. Mice immunized with tyvelose-BSA produce IgG1 antibodies to tyvelose but are not resistant to infection by T. spiralis. Tyvelose-specific antibodies (2.5 mg/20 g) administered to rat pu...
T75536 Koshidacin B

Koshidacin B为针对疟原虫的环四肽类化合物,其针对抗疟原虫(P. falciparum) FCR3和K1系的IC50值分别为0.89 μM与0.83 μM。此化合物在体内能有效抑制疟原虫,适用于疟疾感染的科学研究。
T72519 Niclosamide sodium

BAY2353 sodium

Niclosamide (BAY2353) sodium 为用于研究寄生虫感染的口服抗蠕虫化合物,同时是STAT3抑制剂,在HeLa细胞中IC50为0.25μM。此化合物显示抗癌生物活性,并可抑制Vero E6细胞DNA复制。

化合物

Pyrantel tartrate
Cat.No: T0395
Synonym: Banminth,酒石酸噻吩嘧啶
Target: Antibiotic, Parasite
Pyrantel pamoate
Cat.No: T1259
Synonym: 双羟萘酸噻嘧啶,Pyrantel embonate
Target: Others, Antibiotic, Parasite
Tyvelose
Cat.No: T37757
Synonym:
Target:
Koshidacin B
Cat.No: T75536
Synonym:
Target:
Niclosamide sodium
Cat.No: T72519
Synonym: BAY2353 sodium
Target:
Cat. No. Product Name Target Signaling Pathways
T1104 Paromomycin Sulfate

Aminosidine sulfate,Paromomycin sulfate salt,硫酸巴龙霉素,巴龙霉素硫酸盐

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Paromomycin Sulfate (Aminosidine sulfate) 是一种广谱氨基糖苷类抗生素 ,是具有杀螨杀菌作用的新霉素衍生物。它通过与细菌 30S 核糖体 A 位点的 RNA 寡核苷酸特异性结合,使 mRNA 的翻译提前终止,并抑制蛋白质合成。它可研究细菌和寄生虫感染。

天然产物

Paromomycin Sulfate
Cat.No: T1104
Synonym: Aminosidine sulfate,Paromomycin sulfate salt,硫酸巴龙霉素,巴龙霉素硫酸盐
Target: Antibacterial, Antibiotic, Parasite
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